黄体制剂
黄体制剂（英語：Progestin）是一种合成的[1]孕激素，与孕酮有类似效果。[2]Progestin的两种最重要用途为激素避孕（独立或与雌激素一同使用）以及作为激素替代疗法预防不受对抗的雌激素导致的子宫内膜增生。
参见
参考
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黃體素
（及黄体制剂） | | 孕酮衍生物 | |
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| 逆孕酮衍生物 | |
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17α-羟孕酮衍生物
(and closely related) |
- Acetomepregenol (mepregenol diacetate)
- Algestone
- Algestone acetophenide
- Anagestone acetate
- Chlormadinone acetate
- 醋酸环丙孕酮
- Delmadinone acetate
- Flugestone acetate (flurogestone acetate)
- Hydroxyprogesterone
- Hydroxyprogesterone acetate
- Hydroxyprogesterone caproate
- Hydroxyprogesterone heptanoate
- Medroxyprogesterone
- Medroxyprogesterone acetate#
- Megestrol acetate
- Melengestrol acetate
- Osaterone acetate
- Pentagestrone acetate
- Other 17α-substitutions: Haloprogesterone
- Medrogestone
- Proligestone
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19-去甲孕酮衍生物
(incl. 17α-substituted) |
- Demegestone
- Gestonorone caproate (gestronol hexanoate)
- Nomegestrol acetate
- Norgestomet
- Promegestone
- Segesterone acetate (nestorone)
- Trimegestone
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| 17α-乙炔基睾酮衍生物 | |
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| 19-去甲睾酮衍生物 |
- Estranes: Etynodiol diacetate
- 孕三烯酮
- Lynestrenol
- 炔诺酮#
- 醋酸炔诺酮
- 庚酸炔诺酮
- 异炔诺酮
- Norgestrienone
- Quingestanol acetate
- 替勃龙
- 性腺：去氧孕烯
- Dienogest
- Etonogestrel
- Gestodene
- 左炔诺孕酮#
- Norelgestromin
- Norgestimate
- Norgestrel
- 其他：Allylestrenol
- Altrenogest
- Norgesterone
- Normethandrone (methylestrenolone)
- Norvinisterone
- Oxendolone
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| 17α-Spirolactosteroid |
- Canrenone
- Drospirenone
- Potassium canrenoate
- 螺内酯
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| 其他 | |
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| SPRMs |
- Asoprisnil†
- Telapristone§
- Ulipristal acetate
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| Antiprogestogens | |
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| PR | | 受體致活劑 | |
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| Mixed (SPRMs) |
- Apigenin
- Asoprisnil
- Asoprisnil ecamate
- Guggulsterone
- 山柰酚
- J1042
- LG-120838
- Naringenin
- PRA-910
- 丁香酸
- Telapristone
- 受體拮抗劑： 美服培酮
- Org-31710
- Org-33628
- Ulipristal acetate
- ZK-137316
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| Antagonists |
- 3α-Hydroxytibolone
- 3β-Hydroxytibolone
- 阿来司酮
- 利洛司酮
- 洛那立生
- 奥那司酮
- 托立司酮
- 丙戊酸
- 维拉立生
- 扎诺特隆
- ZM-150271
- ZM-172406
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mPRs
(PAQRs) | | 受體致活劑 |
- 5α-Dihydroprogesterone
- 5β-Dihydroprogesterone
- 11-脱氧皮质酮
- 17α-Hydroxyprogesterone
- 17α,21-Dihydroxyprogesterone
- Allopregnanolone
- 美服培酮
- 孕烯醇酮
- 孕酮
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| Antagonists | |
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| 雌激素 | ER（雌激素受體）
激動劑 |
- （甾體類） Alfatradiol
- 某些雄激素/合成类固醇(e.g., testosterone, testosterone esters, methyltestosterone, metandienone, nandrolone esters) (via estrogenic metabolites)
- 某些黃體製劑 (例如：諾瑞酮，左炔诺孕酮二醋酸酯，替前列酮)
- 氯米酮
- 醋酸邻雌二醇
- 共轭雌三醇
- 共轭雌激素
- 环雌三醇
- 环雌甲酮
- 酯化雌激素
- 雌四醇†
- 雌二醇
- Estradiol esters (e.g., estradiol acetate, estradiol benzoate, estradiol cypionate, estradiol enanthate, estradiol undecylate, estradiol valerate, polyestradiol phosphate, estradiol ester mixtures (Climacteron))
- Estramustine phosphate
- Estriol
- Estriol esters (e.g., estriol succinate, polyestriol phosphate)
- Estrogenic substances
- Estrone
- Estrone esters
- * Estrone sulfate
- * Estropipate (piperazine estrone sulfate)
- Ethinylestradiol#
- * Ethinylestradiol sulfonate
- Hydroxyestrone diacetate
- Mestranol
- Methylestradiol
- Moxestrol
- Nilestriol
- Prasterone (dehydroepiandrosterone; DHEA)
- Prasterone enanthate
- Prasterone sulfate
- Promestriene
- Quinestradol
- Quinestrol
- （非甾體類） Benzestrol
- Bifluranol
- Chlorotrianisene
- Dienestrol
- 双乙酸双烯雌酚
- 乙烯雌酚（己烯雌酚(stilbestrol)）
- Diethylstilbestrol esters/ethers
- Dimestrol (diethylstilbestrol dimethyl ether)
- Fosfestrol (diethylstilbestrol diphosphate)
- Mestilbol (diethylstilbestrol monomethyl ether)
- Doisynoestrol (fenocycline)
- Hexestrol
- Hexestrol esters
- Methallenestril
- Methestrol (promethestrol)
- Methestrol dipropionate (promethestrol dipropionate)
- Paroxypropione
- Quadrosilan
- Triphenylbromoethylene
- Triphenylchloroethylene
- Zeranol
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| 促性腺激素 | |
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| 抗雌激素 | ER拮抗剂
(包含SERMs/SERDs) |
- 异炔诺酮†
- 阿诺尔定
- 贝那普利
- 溴丙雌酚
- 可洛米芬#
- 环苯基酚
- 左旋氯米芬†
- 依匹替司醇
- 拉索瑞烯
- 美匹替坦
- 奥美洛昔芬
- 奥司贝麦芬
- 雷洛昔芬
- 他莫昔芬#
- 托瑞米芬
- （完全抗性的） 依瑞雌苷
- 氟維司群
- （不完全抗性的） 曲洛司坦
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| 芳香酶抑制剂 | |
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| 抗性腺激素 |
- 雄激素/合成類固酮 (例如 睪酮, 睪酮酯, nandrolone esters, oxandrolone, 氟氧孕酮)
- D2 receptor antagonists (prolactin releasers) (e.g., domperidone, metoclopramide, risperidone, haloperidol, chlorpromazine, sulpiride)
- GnRH agonists (e.g., leuprorelin, goserelin)
- GnRH antagonists (e.g., cetrorelix, elagolix)
- Progestogens (e.g., chlormadinone acetate, cyproterone acetate, gestonorone caproate, hydroxyprogesterone caproate, medroxyprogesterone acetate, megestrol acetate)
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| 其他 |
- 混合作用机制:Danazol
- Gestrinone
- 雄烯二酮抗原: Androvax(雄烯二酮白蛋白)
- Ovandrotone albumin (Fecundin)
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- 參見
- 雌激素受体调节剂（模板）
- 雄激素和抗雄激素（模板）
- 孕激素和抗孕激素（模板）
- 雌激素列表
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黃體素
（及黄体制剂） | | 孕酮衍生物 | |
|---|
| 逆孕酮衍生物 | |
|---|
17α-羟孕酮衍生物
(and closely related) |
- Acetomepregenol (mepregenol diacetate)
- Algestone
- Algestone acetophenide
- Anagestone acetate
- Chlormadinone acetate
- 醋酸环丙孕酮
- Delmadinone acetate
- Flugestone acetate (flurogestone acetate)
- Hydroxyprogesterone
- Hydroxyprogesterone acetate
- Hydroxyprogesterone caproate
- Hydroxyprogesterone heptanoate
- Medroxyprogesterone
- Medroxyprogesterone acetate#
- Megestrol acetate
- Melengestrol acetate
- Osaterone acetate
- Pentagestrone acetate
- Other 17α-substitutions: Haloprogesterone
- Medrogestone
- Proligestone
|
|---|
19-去甲孕酮衍生物
(incl. 17α-substituted) |
- Demegestone
- Gestonorone caproate (gestronol hexanoate)
- Nomegestrol acetate
- Norgestomet
- Promegestone
- Segesterone acetate (nestorone)
- Trimegestone
|
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| 17α-乙炔基睾酮衍生物 | |
|---|
| 19-去甲睾酮衍生物 |
- Estranes: Etynodiol diacetate
- 孕三烯酮
- Lynestrenol
- 炔诺酮#
- 醋酸炔诺酮
- 庚酸炔诺酮
- 异炔诺酮
- Norgestrienone
- Quingestanol acetate
- 替勃龙
- 性腺：去氧孕烯
- Dienogest
- Etonogestrel
- Gestodene
- 左炔诺孕酮#
- Norelgestromin
- Norgestimate
- Norgestrel
- 其他：Allylestrenol
- Altrenogest
- Norgesterone
- Normethandrone (methylestrenolone)
- Norvinisterone
- Oxendolone
|
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| 17α-Spirolactosteroid |
- Canrenone
- Drospirenone
- Potassium canrenoate
- 螺内酯
|
|---|
| 其他 | |
|---|
|
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| SPRMs |
- Asoprisnil†
- Telapristone§
- Ulipristal acetate
|
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| Antiprogestogens | |
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|