Template:雄激素类和抗雄激素类
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激动药 | |
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抗雄激素 | AR受体拮抗剂 |
- 甾体类: Abiraterone acetate +niraparib
- Canrenone
- Chlormadinone acetate
- 醋酸环丙孕酮
- Delmadinone acetate
- Dienogest
- Drospirenone
- Medrogestone
- Megestrol acetate
- Nomegestrol acetate
- Osaterone acetate
- Oxendolone
- Potassium canrenoate
- 螺内酯
- 非甾体类: Apalutamide
- Bicalutamide
- 西咪替丁
- Darolutamide
- Enzalutamide
- 氟他胺
- Ketoconazole
- Nilutamide
- Seviteronel†
- Topilutamide (fluridil)
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类固醇生成抑制剂 | 5α-还原酶 |
- Alfatradiol
- Dutasteride
- Epristeride
- Finasteride
- Saw palmetto extract
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其它 |
- Abiraterone acetate +niraparib
- Aminoglutethimide
- Bifluranol
- 醋酸环丙孕酮
- 氟他胺
- Ketoconazole
- Nilutamide
- Seviteronel†
- 螺内酯
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抗促性腺激素 |
- D2 receptor antagonists (prolactin releasers) (e.g., domperidone, 甲氧氯普胺, risperidone, haloperidol, 氯丙嗪, sulpiride)
- Estrogens (e.g., bifluranol, 己烯雌酚, 雌二醇, estradiol esters, ethinylestradiol, ethinylestradiol sulfonate, paroxypropione)
- GnRH agonists (e.g., leuprorelin)
- GnRH antagonists (e.g., cetrorelix)
- Progestogens (incl., chlormadinone acetate, 醋酸环丙孕酮, hydroxyprogesterone caproate, gestonorone caproate, medroxyprogesterone acetate, megestrol acetate)
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其它 |
- 雄烯二酮免疫剂: Androvax (androstenedione albumin)
- Ovandrotone albumin (Fecundin)
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